X-Ceptor Therapeutics

San Diego, United States Founded: 1999 • Age: 27 yrs Acquired By Exelixis
Nuclear receptor modulating small molecule drugs for metabolism and cardiovascular diseases

About X-Ceptor Therapeutics

X-Ceptor Therapeutics is a Healthcare company based in San Diego (United States) founded in 1999, and was acquired by Exelixis in September 2004. Nuclear receptor modulating small molecule drugs for metabolism and cardiovascular diseases. Its focus areas include Life Sciences, Cardiac and Vascular Disorders, Drugs and Diversified. Its competitors include Portola Pharma, MyoKardia and Cellino; 3 of its 3 listed competitors have raised funding.

Company details

X-Ceptor Therapeutics was founded in 1999 in San Diego, United States, and operated in the biotechnology sector. Small molecule therapeutics were developed to modulate nuclear receptors linked to cholesterol metabolism and cardiovascular conditions. A reverse endocrinology method was employed to validate targets, establish disease proof-of-concept, and advance preclinical candidates. The company was acquired by Exelixis in September 2004 for 22.3 million in cash and stock.

  • Headquarters San Diego, United States
  • Stage Acquired
  • Sectors
    Healthcare
  • Website x-ceptor.com
  • Acquired by Exelixis (Sep 2004)
Key Metrics

Funding Insights of X-Ceptor Therapeutics

  • Total Rounds 2
  • Investors Count 3

All 2 funding rounds of X-Ceptor Therapeutics with amounts and investors; the two latest post-money valuations are shown, the rest are part of the premium plan.

DateAmountTransaction NameValuationLead InvestorsInvestors
Oct 1999Series B––
Jun 1999Series B––
Valuation history

4 investors in total: 4 institutional.

Investors in X-Ceptor Therapeutics

X-Ceptor Therapeutics has secured backing from 4 investors, including institutional and venture fund investors. Prominent investors backing the company include Exelixis, Ligand Pharmaceuticals and Farallon Capital Management.

All
Venture Fund
Institutional
InvestorDescriptionFounded YearDomainLocation
Private equity firm
1980gimv.comAntwerp, Belgium
Multiple investment strategies are pursued by this hedge fund.
1986faralloncapital.comSan Francisco, United States
Pharmaceutical drugs are manufactured and developed in the United States.
1987ligand.comSan Diego, United States
Small molecule drugs for cancer treatment are developed.
1994exelixis.comSan Francisco, United States
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Investor details for X-Ceptor Therapeutics

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Timeline of X-Ceptor Therapeutics

4 dated milestones of X-Ceptor Therapeutics across 5 years, from founding to its latest funding, stage changes and deals.

  1. Founded X-Ceptor Therapeutics is founded.
  2. Funding First funding round.
  3. Funding Latest funding round, Series B,.
  4. Exit Acquired by Exelixis.

Competitors of X-Ceptor Therapeutics

X-Ceptor Therapeutics has 3 listed competitors in our database, 3 of them funded. They include Portola Pharma, MyoKardia and Cellino.

Company NameDomainFoundedHQ LocationTotal fundingEmployeesDescription
portola.com2003San Francisco, United States$296.09M369
Therapeutics for cardiovascular and autoimmune diseases are developed.
myokardia.com2012San Francisco, United States$98M224
Specialized drugs are developed for genetic heart diseases.
cellinobio.com2017Cambridge, United States$125M63
Developer of autologous cell therapies
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Detailed competitors of X-Ceptor Therapeutics

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Top companies in Cardiac and Vascular Disorders

3 companies that operate in the same segment as X-Ceptor Therapeutics (Cardiac and Vascular Disorders) in United States, ranked by their profile score on The Company Check.

CompanyDescriptionFoundedLocationTotal fundingRevenueEmployees
Gene-editing therapies for coronary artery disease are developed.
2018Cambridge, Massachusetts, United StatesUSD 215.5 M255
Cardiac monitoring devices and applications are provided for heart health.
2010Mountain View, California, United StatesUSD 114.38 MUSD 6.18 M67
Therapies for lowering low-density lipoprotein cholesterol levels are developed.
1998Ann Arbor, Michigan, United StatesUSD 129.7 MUSD 332.31 M304
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Related news about X-Ceptor Therapeutics

Exelixis to buy X-Ceptor Therapeutics for $22.3M
Marketwatch β€’ 22 years ago
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Complete news archive for X-Ceptor Therapeutics

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Frequently Asked Questions about X-Ceptor Therapeutics

X-Ceptor Therapeutics was founded in 1999.

X-Ceptor Therapeutics is headquartered in San Diego, United States. It is registered at San Diego, California, United States.

X-Ceptor Therapeutics was founded in 1999 in San Diego, United States, and operated in the biotechnology sector. Small molecule therapeutics were developed to modulate nuclear receptors linked to cholesterol metabolism and cardiovascular conditions. A reverse endocrinology method was employed to validate targets, establish disease proof-of-concept, and advance preclinical candidates. The company was acquired by Exelixis in September 2004 for 22.3 million in cash and stock.

X-Ceptor Therapeutics's top competitors include Cellino, MyoKardia and Portola Pharma.

X-Ceptor Therapeutics has 4 investors. Key investors include Exelixis, Ligand Pharmaceuticals, Farallon Capital Management, and Gimv.

Yes. X-Ceptor Therapeutics was acquired by Exelixis in September 2004.

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